产品名称

EMPA

产品货号

Axon 2012 CAS [680590-49-2] MF C23H26N4O4SMW 454.54 Purity: 99% Soluble in DMSO and Ethanol Description Highly potent and selective orexin type 2 (OX2) receptor antagonist, with Ki values of >900 and 1 nM for OX1 and OX2 receptors respectively References Certificates Categories Extra info P Malherbe et al. Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX2 receptor. Br. J. Pharmacol. 2009, 156, 1326–1341. TE Scammell and CJ Winrow. Orexin Receptors: Pharmacology and Therapeutic Opportunities. Annu. Rev. Pharmacol. Toxicol. 2011. 51:243–66. Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology CNS Diabetes & Metabolism Endocrinology A6 Orexin (OX) Orexin type 2 (OX2) receptor antagonist Chemical name N-ethyl-2-(N-(6-methoxypyridin-3-yl)-2-methylphenylsulfonamido)-N-(pyridin-3-ylmethyl)acetamide Parent CAS No. [680590-49-2] Order Size Unit Price Stock 10 mg €135.00 In Stock

产品价格

现货询价，电话：010-67529703

产品规格

产品品牌

axonmedchem

产品概述

产品详情

EMPA

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 2012

CAS [680590-49-2]

MF C23H26N4O4S
MW 454.54

Purity: 99%
Soluble in DMSO and Ethanol

EMPA

Description

Highly potent and selective orexin type 2 (OX2) receptor antagonist, with Ki values of >900 and 1 nM for OX1 and OX2 receptors respectively

P Malherbe et al. Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX2 receptor. Br. J. Pharmacol. 2009, 156, 1326–1341.

TE Scammell and CJ Winrow. Orexin Receptors: Pharmacology and Therapeutic Opportunities. Annu. Rev. Pharmacol. Toxicol. 2011. 51:243–66.

Orexin type 2 (OX2) receptor antagonist

Chemical name

N-ethyl-2-(N-(6-methoxypyridin-3-yl)-2-methylphenylsulfonamido)-N-(pyridin-3-ylmethyl)acetamide

Parent CAS No.

[680590-49-2]

产品资料