产品名称

NCRW0005-F05

产品货号

Axon 2609 CAS [342779-66-2] MF C16H13F2NO2MW 289.28 Purity: 99% Soluble in DMSO Description First antagonist selective for GPR139 (IC50 value 0.21 µM); a useful tool to study GPR139 pharmacology, especially in combination with the GPR139 agonist JNJ 63533054 (Axon 2569) KEYWORDS: NCRW0005-F05 | supplier | GPR139 antagonist | NCRW0005F05 | CAS [342779-66-2] | GPR139 | GPCR | orphan | CNS | Gαq | G-alphaq | diabetes | obesity | Parkinson’s

产品价格

现货询价，电话：010-67529703

产品规格

产品品牌

axonmedchem

产品概述

产品详情

NCRW0005-F05

Based on 1 reference(s) in Google Scholar 9 10 1

Axon 2609

CAS [342779-66-2]

MF C16H13F2NO2
MW 289.28

Purity: 99%
Soluble in DMSO

NCRW0005-F05

Description

First antagonist selective for GPR139 (IC50 value 0.21 µM); a useful tool to study GPR139 pharmacology, especially in combination with the GPR139 agonist JNJ 63533054 (Axon 2569)

KEYWORDS: NCRW0005-F05 | supplier | GPR139 antagonist | NCRW0005F05 | CAS [342779-66-2] | GPR139 | GPCR | orphan | CNS | Gαq | G-alphaq | diabetes | obesity | Parkinson’s

J Wang et al. High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139. Acta Pharmacol Sin. 2015 Jul;36(7):874-8.

CNS Diabetes & Metabolism Miscellaneous Unclassified GPR139

GPR139 antagonist; useful tool to study GPR139 pharmacology

Chemical name

3,3-difluoro-4-(4-methoxyphenyl)-1-phenylazetidin-2-one

Parent CAS No.

[342779-66-2]

产品资料