| 产品详情 |
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| Product Name | Enzastaurin |
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| Description | Purity >98%. Enzastaurin is a potent inhibitor of PKCBeta (IC50 = 6 nM), with modest selectivity over PKCAlpha, PKCGamma, and PKCe (IC50 = 39, 83, and 110 nM, respectively). At 3 µM, enzastaurin also inhibits signaling through the Akt pathway. It suppresses angiogenesis, induces apoptosis, and reduces proliferation of cultured tumor cells. Because of these effects, enzastaurin has potential antineoplastic activity. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 3-(1-methyl-1H-indol-3-yl)-4-[1-[1-(2-pyridinylmethyl)-4-piperidinyl]-1H-indol-3-yl]-1H-pyrrole-2,5-dione, LY317615 |
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| Gene, Accession, CAS # | CAS: 170364-57-5 |
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| Catalog # | LS-H7675 |
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| Price | |
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| Order / More Info | Enzastaurin from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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