产品名称 Tyrphostin SU 1498 ((E)-N-(3?-Phenylpropyl)-α-cyano-3?,5?-diisopropyl-4?-hydroxycinnamamide) from UNITED STATES BIOLOGICAL
产品货号 T9250-80
产品价格 现货询价,电话:010-67529703
产品规格 1mg
产品品牌 UNITED STATES BIOLOGICAL
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Product NameTyrphostin SU 1498 ((E)-N-(3?-Phenylpropyl)-α-cyano-3?,5?-diisopropyl-4?-hydroxycinnamamide)
DescriptionPurity ~98% (TLC). A potent and selective inhibitor (IC50=700nM) of vascular endothelial growth factor receptor 2 (VEGFR 2) (also known as Flk1). Very weak inhibitor of PDGFR-kinase (IC50 >50uM), EGFR-kinase (IC50 >100uM) and HER-2 kinase (IC50>100uM). SU1498 has been shown to cause accumulation of phosphorylated ERK and inhibits its activity in vivo and in vitro by inhibition of ERK dephosphorylation. Solubility: DMSO (~20mg/ml) Molecular Weight: ~390.52
Size1mg
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Catalog #T9250-80
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Order / More InfoTyrphostin SU 1498 ((E)-N-(3?-Phenylpropyl)-α-cyano-3?,5?-diisopropyl-4?-hydroxycinnamamide) from UNITED STATES BIOLOGICAL
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