| 产品详情 |
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| Product Name | Ro3280 |
| Description | Purity ≥98%. Ro3280 is a Polo-like kinase 1 (PLK1) inhibitor. Ro3280 shows strong antitumor activity in xenograft mouse models, has good selectivity against other kinases and has excellent in vitro cellular potency. Synonyms: 4-((9-Cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide; 4-[(9-Cyclopentyl-7,7-difluoro-6,7,8,9-tetrahydro-5-methyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide CAS Number: 1062243-51-9 Molecular Formula: CHFNO Molecular Weight: 543.61 Purity: 98+% Solubility: Alcohol: 100 mg/mL (183.95 mM); DMSO: 100 mg/mL (183.95 mM); Water: Insoluble |
| Size | 5mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 4-((9-Cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide; 4-[(9-Cyclopentyl-7,7-difluoro-6,7,8,9-tetrahydro-5-methyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide |
| Gene, Accession, CAS # | CAS: 1062243-51-9 |
| Catalog # | 380363 |
| Price | |
| Order / More Info | Ro3280 from UNITED STATES BIOLOGICAL |
| Product Specific References | n/a |
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