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| Product Name | BAG 956 |
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| Description | Dual PDPK1 (PDK1) and class I PI 3-K inhibitor (IC50 values are 245, 56, 446, 35 and 117 nM for PDPK1 and PI 3-K p110 -α, -β, -δ, and -γ respectively). Inhibits cellular AKT phosphorylation at Thr308. Blocks cell proliferation, causing arrest in G1 phase of the cell cycle. Slows tumor progression in mouse xenograft models. Purity 99%. MW (observed): 427.5 |
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| Size | 50 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyridinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-benzeneacetonitrile |
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| Gene, Accession, CAS # | CAS: 853910-02-8 |
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| Catalog # | 3606/50 |
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| Price | |
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| Order / More Info | BAG 956 from TOCRIS BIOSCIENCE
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| Product Specific References | n/a |
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| 产品资料 |
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