| 产品详情 |
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| Product Name | Arachidonoyl-2'-Fluoroethylamide |
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| Description | Purity >98%. Arachidonoyl-2'-fluoroethylamide (2-fluoro AEA) is an analog of anandamide in which the alcohol of the ethanolamide group has been removed and replaced with a fluorine atom. This substitution adds considerably increased binding affinity for the CB1 receptor (Ki s = 26.7 and 908 nM for CB1 and CB2, respectively). It also contributes additional selectivity, in that binding to CB2 is decreased relative to AEA. However, the in vivo activity of 2-fluoro AEA is enhanced much less than the binding affinity, because the analog remains a good substrate for FAAH and is rapidly hydrolyzed by this enzyme. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-(2-fluoroethyl)-5Z,8Z,11Z,14Z-eicosatetraenamide, 2'-fluoro AEA, 2'-fluoro Anandamide |
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| Gene, Accession, CAS # | CAS: 166100-37-4 |
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| Catalog # | LS-H6601 |
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| Order / More Info | Arachidonoyl-2'-Fluoroethylamide from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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