| 产品详情 |
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| Product Name | Mepyramine (maleate) |
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| Description | Purity >95%. Mepyramine is a first generation antihistamine that acts as an inverse agonist at the histamine H1 receptor. It is reported to bind with high affinity to a Gq/11 protein-coupled form of the receptor and to promote a G protein-coupled inactive state of the H1 receptor that interferes with the Gq/11 -mediated signaling of the endogenously expressed receptor, as well as to reduce G protein availability for other non-related receptors associated with this signaling pathway. Mepyramine has been shown to inhibit histamine-induced inositol phosphate production with a log EC50 value of -7.94. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N1 -[(4-methoxyphenyl)methyl]-N2 ,N2 -dimethyl-N1 -2-pyridinyl-1,2-ethanediamine, 2Z-butenedioate, NSC 3604, Pyrilamine |
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| Gene, Accession, CAS # | CAS: 59-33-6 |
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| Catalog # | LS-H8637 |
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| Order / More Info | Mepyramine (maleate) from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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