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| Product Name | Efaroxan hydrochloride |
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| Description | Purity >98% by HPLC. Potent and highly selective a-2 adrenoceptor antagonist and imidazoline I1 receptor ligand (Ki values are 13.5, 38, 1820, 52.5 and < 10000 nM for a-2A, a-2B, a-2C, I1, and I2 receptors respectively). Like several other imidazoline reagents, it elicits a glucose-dependent increase in insulin secretion from pancreatic Beta-cells. This response has been attributed to efaroxan-mediated blockade of KATP channels, with the subsequent gating of voltage-sensitive calcium channels. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 2-(2-Ethyl-2,3-dihydro-2-benzofuranyl)-4,5-dihydro-1H-imidazole hydrochloride |
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| Gene, Accession, CAS # | CAS: 88917-00-2 |
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| Catalog # | LS-H10801 |
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| Order / More Info | Efaroxan hydrochloride from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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