产品名称 Barnidipine (hydrochloride) from LIFESPAN BIOSCIENCES INC.
产品货号 LS-H6739
产品价格 现货询价,电话:010-67529703
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产品品牌 LIFESPAN BIOSCIENCES INC.
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Product NameBarnidipine (hydrochloride)
DescriptionPurity >98%. Barnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery. It demonstrates antihypertensive activity by reducing peripheral vascular resistance. It decreases blood pressure in spontaneously hypertensive rats when administered orally at 1 and 3 mg/kg per day. Formulations containing barnidipine have been used as a treatment for hypertension. In obstructive sleep apnea patients with non-dipper pattern hypertension, barnidipine reduced mean nighttime systolic and diastolic arterial blood pressure.
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Other Names(4S)-3,5-pyridinedicarboxylic acid, 3-methyl 5-[(3S)-1-(phenylmethyl)-3-pyrrolidinyl] ester, monohydrochloride, YM-09730-5
Gene, Accession, CAS #CAS: 104757-53-1
Catalog #LS-H6739
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Order / More InfoBarnidipine (hydrochloride) from LIFESPAN BIOSCIENCES INC.
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