| 产品详情 |
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| Product Name | CCG-50014 |
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| Description | Purity >98%. CCG-50014 is an inhibitor of regulator of G protein signaling 4 (RGS4) (IC50 = 30 nM) and is > 20-fold selective for RGS4 over other RGS proteins. RGS proteins bind to the GAlpha subunits of activated heterotrimeric G proteins and accelerate the rate of GTP hydrolysis, acting as GTPase-activating proteins. CCG-50014 irreversibly binds and destabilizes RGS4 with no effect on GAlpha0, while blocking GTPase activity and GAlpha0 -dependent translocation of RGS4 to the membrane. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 4-[(4-fluorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione |
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| Gene, Accession, CAS # | CAS: 883050-24-6 |
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| Catalog # | LS-H7029 |
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| Price | |
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| Order / More Info | CCG-50014 from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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