产品名称 TCS-OX2-29 from LIFESPAN BIOSCIENCES INC.
产品货号 LS-H10132
产品价格 现货询价,电话:010-67529703
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产品品牌 LIFESPAN BIOSCIENCES INC.
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Product NameTCS-OX2-29
DescriptionPurity >98%. Orexin receptors R1 (OX1R) and OX2R mediate the action of the neuropeptides orexin A and orexin B. TCX-OX2-29 is an antagonist of OX2R (pKi = 7.5) that exhibits >250-fold selectivity for hOX2R compared with hOX1R (IC50 s = 40 nM and >10,000 nM, respectively). It blocks the inhibitory action of orexin A on forskolin-induced cAMP formation.
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Other Names(2S)-1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-1-butanone, monohydrochloride
Gene, Accession, CAS #CAS: 1610882-30-8
Catalog #LS-H10132
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Order / More InfoTCS-OX2-29 from LIFESPAN BIOSCIENCES INC.
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