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| Product Name | GSK-1016790A |
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| Description | Purity >98% by NMR, TLC. GSK-1016790A is a novel and potent TRPV4 channel agonist. GSK-1016790A induced Ca2+ influx in mouse and human TRPV4 expressing HEK cells (EC50 values of 18 and 2.1 nM, respectively), and evoked a dose-dependent activation of TRPV4 whole-cell currents at concentrations above 1 nM. It is 300-fold more potent than 4a-PDD and is a valuable tool for investigating the role of TRPV4 in physiological processes. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | (N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide |
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| Gene, Accession, CAS # | CAS: 942206-85-1 |
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| Catalog # | LS-H14694 |
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| Order / More Info | GSK-1016790A from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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